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Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
This page covers what the list does and does not say about 5-Amino-1MQ, how the S0 catch-all works, what that means in practice for tested athletes, how college sport treats unlisted compounds, what a workplace drug test looks for, and where 5-Amino-1MQ stands with the FDA. It is general information, not anti-doping advice. For the compound itself, read what is 5-Amino-1MQ.
5-Amino-1MQ is not named on the 2026 WADA Prohibited List, but a tested athlete should not read that as permission. The list's S0 class prohibits, at all times, any pharmacological substance not addressed elsewhere on the list that has no current approval by any governmental health authority for human therapeutic use, and 5-Amino-1MQ is not approved for anything. WADA's own explanatory note warns that a substance not specifically named "may still be prohibited." The FUSION blend that contains it is prohibited outright, because it also contains MOTS-c, BPC-157 and tesamorelin.
This page covers what the list does and does not say about 5-Amino-1MQ, how the S0 catch-all works, what that means in practice for tested athletes, how college sport treats unlisted compounds, what a workplace drug test looks for, and where 5-Amino-1MQ stands with the FDA. It is general information, not anti-doping advice. For the compound itself, read what is 5-Amino-1MQ.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
The short answer
| The question | The answer | What to do |
|---|---|---|
| Is 5-Amino-1MQ named on the 2026 WADA List? | No. The live pages do not find it named | Do not stop there |
| Could it still be prohibited? | Yes. S0 covers unapproved pharmacological substances that are not named, and WADA warns unnamed substances may still be prohibited | Check Global DRO and ask your anti-doping body |
| Is it approved anywhere for human use? | The live record describes it as not approved for anything | This is the condition S0 is written around |
| Is the FUSION blend prohibited? | Yes. It contains MOTS-c (S4.4.1), BPC-157 (S0) and tesamorelin (S2.2.4) | Do not use it if tested |
| Will it show up on a workplace drug test? | No. Workplace panels screen for drugs of abuse only | Nothing to do |
| Does a prescription protect me? | No. Anti-doping runs on strict liability | Only an advance therapeutic use exemption does |
The honest summary: nobody can tell you from a web page that 5-Amino-1MQ is permitted, and the structure of the list leans the other way.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
What 5-Amino-1MQ is, and why that matters here
5-Amino-1MQ is not a peptide. It is a small synthetic molecule, a methylquinolinium compound, designed to inhibit an enzyme called nicotinamide N-methyltransferase (NNMT). The full explanation is in is 5-Amino-1MQ a peptide. It is prescribed alongside peptides because it is compounded and dispensed the same way.
That matters for anti-doping in one specific way. People sometimes assume that because WADA's peptide rules are about hormones and growth factors, a small molecule falls outside them. It does not work like that. S0 is not about peptides at all: it covers any pharmacological substance, of any structure, that meets its conditions.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
How the S0 catch-all works
The wording
S0, Non-Approved Substances, prohibits at all times "any pharmacological substance which is not addressed by any of the subsequent sections of the List and with no current approval by any governmental regulatory health authority for human therapeutic use." The 2026 List gives examples, BPC-157 among them, alongside 2,4-dinitrophenol, ryanodine receptor-1-calstabin complex stabilizers and troponin activators. The list describes the class as drugs in development, discontinued drugs, designer drugs and veterinary-only substances.
Why it prohibits things it does not name
S0 catches substances by regulatory status rather than by name. A substance need not appear on the list at all; it only needs to lack regulatory approval for human therapeutic use and not be captured by another section. That is the most important clause for anyone looking up an unlisted compound.
WADA's own note on unnamed substances
The 2027 List's explanatory note puts it directly: "Many peptides, not approved for human use by regulatory authorities, fulfill the criteria of the World Anti-Doping Code for inclusion on the Prohibited List and fall under the S0 (Non-Approved Substances) class, or other classes (such as S2 or S4). Even if a peptide is not specifically named on the List, utmost caution should be taken as it may still be prohibited." 5-Amino-1MQ is not a peptide, but S0's wording covers any pharmacological substance, so the same caution applies.
Where 5-Amino-1MQ sits against that test
S0 condition 5-Amino-1MQ, on the live record A pharmacological substance Yes: a synthetic enzyme inhibitor prescribed as an injection Not addressed by another section of the List Not named in any section the live pages cite No current approval by any governmental health authority for human therapeutic use Described as not approved for anything; no human trials of any design have been published Whether a given anti-doping body would classify it under S0 is their determination, not this page's. But every condition the clause sets out is one 5-Amino-1MQ appears to meet, which is why the safe reading for a tested athlete is to treat it as off limits unless their anti-doping organisation says otherwise in writing.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
The FUSION blend is not a grey area
FUSION Blend combines BPC-157, MOTS-c, 5-Amino-1MQ and tesamorelin in one 5 mL vial. Whatever the status of 5-Amino-1MQ, three of its four ingredients are prohibited at all times:
| Ingredient in FUSION | Where it sits on the 2026 List |
|---|---|
| BPC-157 | S0, named explicitly as an example |
| MOTS-c | S4.4.1, as an activator of AMP-activated protein kinase |
| Tesamorelin | S2.2.4, growth hormone releasing factors |
| 5-Amino-1MQ | Not named; S0 caution applies |
A blend is prohibited by virtue of its components. FUSION is prohibited for a tested athlete, full stop.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
Related compounds people compare it with
5-Amino-1MQ is often discussed with MOTS-c and SLU-PP-332 as "metabolic" compounds. Their anti-doping positions are clearer than its own, and they show where the list has been heading:
- MOTS-c is named under S4.4.1 as an AMPK activator, prohibited at all times, and a validated plasma test for it was published in 2019.
- SLU-PP-332 falls under WADA's prohibition of exercise mimetics and metabolic modulators, and was added to S4.4 by name for 2027, with detection methods published in 2026.
None of that places 5-Amino-1MQ in S4.4; the live pages do not say it is there. It does show that WADA has been naming metabolic compounds as they appear, and that a compound being unnamed this year says little about next year. The comparison is in MOTS-c vs SLU-PP-332 vs 5-Amino-1MQ.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
College sport and workplace tests
The NCAA
The NCAA bans eight drug classes, including hormone and metabolic modulators, and states that "any substance that is chemically/pharmacologically related to one of the above drug classes, even if it is not listed as an example, is also banned." The school and the student-athlete are both accountable. A college athlete should route the question through their athletics health care provider before starting anything, not after.
A standard workplace panel
A standard pre-employment or workplace drug panel does not look for 5-Amino-1MQ. Those panels screen for a short, fixed list of drugs of abuse written into regulation, and nothing in that system looks for a prescribed therapy. More is in do peptides show up on a drug test.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
Strict liability and exemptions
Anti-doping runs on strict liability: the athlete is responsible for what is in their sample, whatever the intent, the supplier or the label. A valid prescription does not change that. Only a therapeutic use exemption granted in advance does, and it requires a diagnosed condition, no reasonable permitted alternative, and no performance enhancement beyond a return to normal health. For a compound with no human trials and no approved indication, that is a hard case to make. A telehealth prescription is not a TUE, and no prescriber can grant one.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
Where 5-Amino-1MQ stands with the FDA
5-Amino-1MQ is not an FDA-approved drug, is not a component of any FDA-approved drug, and has no USP monograph. It does not appear on the 503A Bulks List, and in the FDA's list updated 14 May 2026 it is in none of the three interim categories. It was not before the Pharmacy Compounding Advisory Committee in July 2026, and the FDA has never published a safety-risk finding about it. It is a compounded, prescription-only medication, and compounded medications are not FDA approved. None of that answers the anti-doping question, which turns on approval for human therapeutic use, not on compounding status.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
If you are not a tested athlete
The anti-doping question does not reach a recreational athlete outside any testing pool. What remains is the evidence: mice and cultured cells, with no human trials of any design, set out in 5-Amino-1MQ benefits and 5-Amino-1MQ side effects.
At Pepti, 5-Amino-1MQ is $219 a month, all-in, covering medication, physician review, refill management and shipping, with no membership fee. It is a 5 mL multi-dose vial at 1 mg/mL (5 mg per vial). The typical printed direction is 0.25 mL (25 units on a U-100 syringe) subcutaneously once daily Monday through Friday, which is 0.25 mg per dose and 20 doses, about four weeks, so refills run every 28 days, one vial per fill. Your physician sets your directions after reviewing your intake, and they are printed on the vial.
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests
Where to get 5-Amino-1MQ prescribed
- Complete a free online intake covering your history, medications and whether you are subject to drug testing in any sport or job.
- A physician licensed in your state reviews it, usually within 24 hours.
- If it is appropriate, a PCAB-accredited, FDA-registered US 503A compounding pharmacy prepares it to that prescription. Lot test results are at /quality/lab-results.
- It ships refrigerated with ice packs, sterile syringes and alcohol prep pads, with directions printed on the vial.
- Your physician stays reachable for questions and side effects.
Step by step: how to get 5-Amino-1MQ prescribed online. Bloodwork is not required for any Pepti treatment. If your physician wants labs for your care, they'll ask through your account.
References
What this is based on.
References
- Neelakantan H, Vance V, Wetzel MD et al.. Selective and membrane-permeable small molecule inhibitors of nicotinamide N-methyltransferase reverse high fat diet-induced obesity in mice · Biochem Pharmacol (2018) · PMID 29155147
- Neelakantan H, Wang HY, Vance V et al.. Structure-Activity Relationship for Small Molecule Inhibitors of Nicotinamide N-Methyltransferase · J Med Chem (2017) · PMID 28548833
- Neelakantan H, Brightwell CR, Graber TG et al.. Small molecule nicotinamide N-methyltransferase inhibitor activates senescent muscle stem cells and improves regenerative capacity of aged skeletal muscle · Biochem Pharmacol (2019) · PMID 30753815
- Babula JJ, Bui D, Stevenson HL, Watowich SJ, Neelakantan H. Nicotinamide N-methyltransferase inhibition mitigates obesity-related metabolic dysfunction · Diabetes Obes Metab (2024) · PMID 39161060
- Dimet-Wiley AL, Latham CM, Brightwell CR et al.. Nicotinamide N-methyltransferase inhibition mimics and boosts exercise-mediated improvements in muscle function in aged mice · Sci Rep (2024) · PMID 38969654
- Dimet-Wiley A, Wu Q, Wiley JT et al.. Reduced calorie diet combined with NNMT inhibition establishes a distinct microbiome in DIO mice · Sci Rep (2022) · PMID 35013352
- Kraus D, Yang Q, Kong D et al.. Nicotinamide N-methyltransferase knockdown protects against diet-induced obesity · Nature (2014) · PMID 24717514
- Kannt A, Pfenninger A, Teichert L et al.. Association of nicotinamide-N-methyltransferase mRNA expression in human adipose tissue and the plasma concentration of its product, 1-methylnicotinamide, with insulin resistance · Diabetologia (2015) · PMID 25596852
Citations are provided for educational purposes. They do not constitute medical advice. Always discuss any peptide protocol with your prescribing physician.
Common questions
Is 5-Amino-1MQ Banned in Sports? WADA, the S0 Catch-All and Drug Tests, answered.
It is not named on the 2026 Prohibited List. But S0 prohibits unapproved pharmacological substances that are not named, and 5-Amino-1MQ is not approved for anything, so a tested athlete should not treat it as permitted.
S0 does not list every substance it covers; it catches substances by regulatory status. Whether an anti-doping body applies it to 5-Amino-1MQ is their call to make, and every condition in the clause appears to be met. Ask your anti-doping organisation.
Not on a standard workplace panel, which screens for drugs of abuse only. On anti-doping testing, the live pages do not describe a published method for 5-Amino-1MQ, but lack of a known test does not make a substance permitted, and stored samples can be reanalysed.
Yes. It contains BPC-157 (S0), MOTS-c (S4.4.1) and tesamorelin (S2.2.4), each prohibited at all times.
No. It is a small synthetic molecule that inhibits the enzyme NNMT. That does not take it outside S0, which covers any pharmacological substance.
It is not named in the NCAA's published examples the live pages cite, but the NCAA bans hormone and metabolic modulators and anything pharmacologically related to a banned class. Ask your athletics health care provider first.
You can apply in advance, but it would be a hard case: there are no human trials and no approved indication, and permitted alternatives exist for the goals it is prescribed around.
Search it on Global DRO for your sport and country, keep the reference number, and if the result is ambiguous, ask your national anti-doping organisation in writing. Peptides for athletes covers the wider rules.
It is prescription-only and compounded by licensed pharmacies to a prescription. It is not FDA approved, and being legal to prescribe is a separate question from being permitted in sport. The free assessment goes to a physician licensed in your state. A consultation does not guarantee a prescription.
Next step
See what a physician recommends for you.
A licensed physician in your state reviews your intake and decides what is appropriate. A consultation does not guarantee a prescription.